I-Galantamine Hydrobromide powder umkhiqizi we-CAS No.: 1953-04-4 98% ubumsulwa min.okwengeza izithako
Amapharamitha womkhiqizo
Igama lomkhiqizo | I-Galantamine Hydrobromide |
Elinye igama | I-Galanthamine hydrobromide; I-Galantamine HBr; I-Galanthamine HBr;(4aS,6R,8aS)-4a,5,9,10,11,12-hexahydro-3-methoxy-11-methyl-6H-Benzofuro[3a,3,2-ef][2]benzazepin- 6-ol, Hydrobromide |
Inombolo ye-CAS. | 1953-04-4 |
Ifomula yamangqamuzana | I-C17H21NO3.HBr |
Isisindo samangqamuzana | 368.27 |
Ubumsulwa | 98.0% |
Ukubukeka | impushana emhlophe ukuya emhlophe |
Ukupakisha | 1kg/bag 10kgs,25kgs/drum |
Isicelo | izidakamizwa ze-nootropic |
Isingeniso somkhiqizo
I-Galantamine hydrobromide iwuhlobo lwe-benzozepine etholakala kuma-bulb nezimbali ze-narcissus, i-osmanthus, noma i-canna.Futhi iyi-oral cholinesterase inhibitor.Njenge-ligand ye-nicotinic acetylcholine receptor, iye yasetshenziswa kabanzi ukuthuthukisa umsebenzi we-neurocognitive.Indima yayo ukuvimbela ngokuncintisana nangokuhlehla i-acetylcholinesterase, ngaleyo ndlela kwandise ukugcwala kwe-acetylcholine.
Lapho ingena egazini, i-galanthamine hydrobromide ingena kalula kuzo zonke izingxenye zomzimba, kuhlanganise nobuchopho.Ibophezela ku-nicotinic acetylcholine receptor, ibangele izinguquko ezihambisanayo futhi ikhulise ukukhululwa kwe-acetylcholine.Isebenza futhi ngokuncintisana nokubuyisela emuva imiphumela ye-cholinesterase inhibitors.Ngokuvimbela i-cholinesterase, ivimbela ukubola kwe-acetylcholine, ngaleyo ndlela ikhulise izinga kanye nobude be-neurotransmitter enamandla.I-Galanthamine iphinde ithuthukise ikhono lokufunda nenkumbulo, ivimbele ukuvuvukala kobuchopho futhi igcine amazinga aphezulu ama-neurotransmitters ngokugcina ubuqotho be-neurons nama-synapses.
Isici
(1) Omunye umphumela obalulekile we-galanthamine hydrobromide ekuthuthukiseni inkumbulo amandla ayo okuthuthukisa ukusebenza kwenkumbulo.Inyusa isivinini sokwakheka kwenkumbulo futhi ithuthukise ukugcinwa kwemininingwane namaqiniso.
(2) Ikhono lokufunda liyathuthukiswa ngokwandisa i-synaptic plasticity kanye neuroplasticity.I-Galanthamine hydrobromide ithinta ngokuqondile noma ngokungaqondile i-neuroplasticity.Ivuselela i-synaptic plasticity ngokwenza kusebenze i-microglia ne-astrocyte.
(3) Kuyasiza ukulala futhi kwandisa ukuphumula.I-Galanthamine ingandisa ubunzima bokwenzeka kokulala ngokuvusa ukunyakaza kwamehlo ngokushesha, ngaleyo ndlela ithuthukise ikhwalithi yokulala.
(4) Thuthukisa ukuvikelwa kwe-antioxidant, i-Galantamine inikeza ukuvikelwa kwe-antioxidant ukulwa nokucindezeleka okwenziwe nge-oxidative okubangelwa ama-radicals mahhala.Ingavikela amangqamuzana obuchopho ekulimaleni kwe-oxidative ukuze kugcinwe ukusebenza kahle kobuchopho.