I-Tianeptine Semisulfate Monohydrate umkhiqizi we-powder CAS No.: 1224690-84-9 98% ubumsulwa min.okwengeza izithako
Amapharamitha womkhiqizo
Igama lomkhiqizo | I-Tianeptine Hemisulfate Monohydrate |
Elinye igama | i-tianeptinesulfate; (Thiazepin-11-ylAmino)HeptanoicAcidSemisulfateMonohydrateTianeptineSemisulfateMonohydrate; 7-[(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoicacidsulfatehydrate(2:1:2); I-Tianeptinehemisulfatemonohydrate(THM); 7- [(3-Chloro-6-methyl-5,5-dioxido-6,11-dihydrodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoicacidsulfatehydrate(2:1:2); Tianeptinehemisulfatehydrate;Thiazepin-11-ylAmino)HeptanoicAcidSemisulfate; I-THM |
Inombolo ye-CAS. | 1224690-84-9 |
Ifomula yamangqamuzana | I-C21H27ClN2O8S2 |
Isisindo samangqamuzana | 535.02 |
Ubumsulwa | 98.0% |
Ukubukeka | I-crystal powder emhlophe |
Isicelo | I-Dietary Supplement Raw Material |
Isingeniso somkhiqizo
I-Tianeptine Hemisulfate Monohydrate iyi-serotonin reuptake inhibitor (SSRI) ekhethiwe kanye nomuthi ocindezelayo.Njenge-antidepressant engeyona yendabuko, indlela yayo yokusebenza ihlukile kuleyo yezidakamizwa zendabuko, ithuthukisa isimo sengqondo nesimo somzwelo ngokuthuthukisa i-synaptic plasticity ye-hippocampal neurons.I-Tianeptine Hemisulfate Monohydrate nayo isetshenziselwa ukwelapha ukukhathazeka nokuphazamiseka kwemizwelo.
I-Tianeptine Hemisulfate Monohydrate isetshenziswa kabanzi ocwaningweni lwezokwelapha, ikakhulukazi ekuthuthukisweni kwama-antidepressants.Iyacwaningwa futhi ukuze isetshenziswe ezifweni ze-neurodeergenerative, ukuphathwa kobuhlungu, nokwelashwa kokulutheka.Ukusebenza kwe-Tianeptine Hemisulfate Monohydrate kuye kwafundwa kabanzi futhi kwaqinisekiswa, futhi kuvunyelwe ukwelashwa kokucindezeleka emazweni amaningi.
Kumele kuqashelwe ukuthi nakuba i-Tianeptine Hemisulfate Monohydrate ifakazelwe ukuthi iyi-antidepressant ephumelelayo ekusetshenzisweni kwemitholampilo, ihlukaniswa njengento elawulwayo kwamanye amazwe, enemikhawulo ekusetshenzisweni nasekudayiseni kwayo.Noma ubani osebenzisa noma othenga i-Tianeptine Hemisulfate Monohydrate kufanele aqaphele imithetho neziqondiso ezifanele ezweni lakubo.
Isici
(1) Indlela yokusebenza eyingqayizivele: I-Tianeptine Hemisulfate Monohydrate iyisithuthukisi esikhethiwe se-serotonin reuptake (SSRE), okusho ukuthi ithuthukisa ukutholwa kabusha kwe-serotonin ebuchosheni, okuholela ekwandeni kwe-synaptic plasticity kanye nokuthuthukiswa kwemizwelo.Le ndlela yokusebenza yehlukile kuma-antidepressants endabuko, ngokuvamile okuyi-serotonin reuptake inhibitors (SSRIs).
(2) Ukuqala kwesenzo esisheshayo: I-Tianeptine Hemisulfate Monohydrate inokuqala okusheshayo kwesenzo, ngezifundo zomtholampilo ezibonisa ukuthuthukiswa kwezimpawu zokucindezeleka ekuqaleni kwesonto elilodwa ngemva kokuqala kokwelashwa.
(3) Ukusebenza kwengqondo okuthuthukisiwe: I-Tianeptine Hemisulfate Monohydrate iboniswe ukuthuthukisa umsebenzi wokuqonda ezigulini ezinezinkinga ezinkulu zokucindezeleka, njengenkumbulo nokunaka.
(4) Amandla okulutha aphansi: Ngokungafani namanye ama-antidepressants, i-Tianeptine Hemisulfate Monohydrate inamandla aphansi okulutha futhi ayibangeli izimpawu zokuhoxa lapho iyekwa.Lokhu kungenxa yokuthi ayibhekiseli ohlelweni lwe-dopamine, oluhlotshaniswa nokulutheka nokuncika.
(5) Ukwelashwa kwezinkinga zokukhathazeka: I-Tianeptine Hemisulfate Monohydrate iboniswe ukuthi inemiphumela yokukhathazeka, okwenza kube ukwelashwa okungaba khona kwezinkinga zokukhathazeka ezifana nokukhathazeka okujwayelekile nokukhathazeka komphakathi.
Izinhlelo zokusebenza
I-Tianeptine Hemisulfate Monohydrate iyikhemikhali yezemithi esetshenziswa kabanzi emikhakheni yezokwelapha neyocwaningo.Njengomuthi oqeda ukucindezeleka, ugunyazwe emazweni amaningi ukuze welaphe ukudangala, ukukhathazeka, ukuphazamiseka kwemizwelo, nezinye izifo ezihlobene.Ngaphezu kwalokho, i-Tianeptine Hemisulfate Monohydrate iye yafundelwa amandla ayo ekwelapheni izifo ze-neurodeergenerative ezifana ne-Alzheimer's, ukuphathwa kobuhlungu, nokwelashwa kokulutheka.
Eminyakeni yamuva, i-Tianeptine Hemisulfate Monohydrate ithole ukuthandwa okwandayo ocwaningweni lwezokwelapha, ikakhulukazi ekuthuthukisweni kwezidakamizwa ezilwa nokucindezeleka.Ngocwaningo olwengeziwe oluqinisekisa imiphumela yalo yokwelapha, amathuba okusetshenziswa kwawo aya ngokuya abonakala.I-Tianeptine Hemisulfate Monohydrate ingase ibe isidakamizwa esinemisebenzi eminingi yokwelapha izifo ezihlukahlukene zezinzwa esikhathini esizayo.
Ngaphezu kwalokho, i-Tianeptine Hemisulfate Monohydrate nayo inokusebenza okungenzeka kwezinye izinkambu.Ucwaningo lwakamuva lubonise ukuthi i-Tianeptine Hemisulfate Monohydrate ingase ibe namandla okwelapha izinkinga ze-neurofunctional zangemuva kokushaywa unhlangothi.Ukwengeza, ezinye izifundo ziphakamisa ukuthi i-Tianeptine Hemisulfate Monohydrate ingaba yinzuzo ezifweni ze-metabolic ezifana nokukhuluphala nesifo sikashukela.