Umkhiqizi wempuphu we-OTR-AC（Ostarine Acetate） 98% ubumsulwa obuncane bezithako zesengezo
Amapharamitha Omkhiqizo
| Igama lomkhiqizo | I-OTR-AC |
| Elinye igama | I-Ostarine Acetate |
| Ifomula yama-molecule | C21H16F3N3O4 |
| Isisindo sama-molecule | 431.36 |
| Ubumsulwa | 98.0% |
| Ukubukeka | Impuphu emhlophe |
| Ukupakisha | 1kg/isikhwama 25kg/isigubhu |
| Isicelo | Thola imisipha futhi ulahlekelwe amafutha |
Isingeniso somkhiqizo
I-OTR-AC, eyaziwa nangokuthi i-MK-2866 Ester, yi-MK-2866 (i-Ostarine) eye yathola i-esterification (inqubo yokuhlanganisa i-organic acid notshwala). Le nqubo yamakhemikhali isetshenziselwa ukwandisa amandla ento ethile nokwandisa ingxenye yokuphila (isikhathi esithathayo ukuze inani lehle liye kuhhafu yenani layo lokuqala). Ngenxa yale nqubo, inguqulo ye-ester ye-ostarine inamandla aphindwe kayishumi okugcina umsebenzi webhayoloji. Lokhu kufeza izinzuzo ezengeziwe, njengenguqulo ye-ester ye-selective androgen receptor modulator (SARM) Ostarin, i-OTR-AC inamandla kakhulu futhi ihlala isikhathi eside. Ngokunamathela kuphrotheni emzimbeni ebizwa ngokuthi i-androgen receptor, ivuselela ukwakheka kwezicubu zemisipha. Lokhu kwandisa ubukhulu bemisipha namandla.
Isici
(1) Ubumsulwa obuphezulu: I-OTR-AC ingathola imikhiqizo yobumsulwa obuphezulu ngezinqubo zokukhiqiza ezicwengekile. Ubumsulwa obuphezulu busho ukutholakala okungcono kwe-bioavailability kanye nokusabela okuncane okubi.
(2) Ukuphepha: I-OTR-AC iwumkhiqizo wemvelo oye wafakazelwa ukuthi uphephile emzimbeni womuntu.
(3) Ukuzinza: I-OTR-AC inozinzo oluhle futhi ingagcina umsebenzi wayo kanye nomphumela ngaphansi kwezimo ezahlukene zokubeka kanye nezimo zokubeka.
Izicelo
I-OTR-AC isebenza njenge-selective androgen receptor modulator (SARM), okusho ukuthi isebenza ngokukhetha ezicutshini zemisipha kanye nezicubu zamathambo emzimbeni ngaphandle kokuthinta ezinye izitho nezicubu. Ithuthukisa imisipha kanye nokusebenza ngokomzimba, isiza ukwandisa imisipha kanye namandla ngenkathi inciphisa okuqukethwe kwamafutha. I-OTR-AC isebenza namanye ama-SARM ukwandisa imisipha kanye namandla ngokuvuselela ukwakheka kwezicubu zemisipha. Ngaphezu kokusiza ukwandisa imisipha, i-OTR-AC itholakale ukuthi yehlisa amafutha omzimba jikelele. I-OTR-AC iyanda ngokuthuthukisa i-lipid metabolism kanye nokuthinta ukukhishwa kwe-adiponectin, i-hormone elawula ukuwohloka kwama-fatty acid Ukuphula amaseli amafutha, i-OTR-AC ingasiza ekukhuthazeni ukwakheka kwamathambo nokuvimbela izifo zamathambo.
