Umkhiqizi wempuphu yeFasoracetam Inombolo ye-CAS: 110958-19-5 Ubumsulwa obungu-99% okungenani bezithako ezengeziwe
Ividiyo Yomkhiqizo
Amapharamitha Omkhiqizo
| Igama lomkhiqizo | I-Fasoracetam |
| Elinye igama | I-FASORACETAM; (5R)-5-(piperidine-1-carbonyl)-2-pyrrolidone; (5R)-5-(piperidine-1-carbonyl)pyrrolidin-2-one; (5R)-5-piperidin-1-ylcarbonylpyrrolidin-2-one |
| Inombolo ye-CAS | 110958-19-5 |
| Ifomula yama-molecule | C10H16N2O2 |
| Isisindo sama-molecule | 196.25 |
| Ubumsulwa | 99.0% |
| Ukubukeka | Impuphu emhlophe ekristalu |
| Ukupakisha | 1 kg/isikhwama 25kg/isigubhu |
| Isicelo | I-Nootropic |
Isingeniso somkhiqizo
I-Fasoracetam, iyinhlanganisela ye-nootropic eyasungulwa okokuqala eJapane. Ifana ngesakhiwo nezinye izinhlobo ze-racemate njenge-piracetam, kodwa ikhombisa izici zesenzo ezihlukile. I-Fasoracetam kucatshangwa ukuthi ilawula imiphumela yama-neurotransmitter ahlukahlukene ebuchosheni, okuhlanganisa nezinhlelo ze-GABA, i-glutamatergic, kanye ne-cholinergic. Ngokuthinta ukukhululwa nokumuncwa kwala ma-neurotransmitter, i-fasoracetam ingathuthukisa imisebenzi yokuqonda njengokunaka, ukuhlanganiswa kwenkumbulo, kanye nokucubungula ulwazi. Ucwaningo kanye nobufakazi obungahleliwe busikisela ukuthi i-fasoracetam inganikeza izinzuzo eziningi zokuqonda. Omunye wemiphumela yayo eyinhloko ukuthuthukisa ukugxilisa ingqondo kanye nesikhathi sokunaka, okwenza kube usizo olungaba khona kulabo abahlushwa yi-attention deficit disorder noma i-attention deficit hyperactivity disorder (ADD/ADHD). Izifundo zokuqala zibonise imiphumela ethembisayo, ezibonisa ikhono le-fasoracetam lokuthuthukisa ukunaka, ukunciphisa ukungaziphathi kahle kanye nokuthuthukisa ukulawula kwengqondo. Ngaphezu kwalokho, izifundo zezilwane zibonisa ukuthi i-Fasoracetam ithuthukisa amandla esikhathi eside, inqubo ehlotshaniswa nokwakheka kwememori kanye ne-synaptic plasticity.
Isici
(1) Ukuhlanzeka okuphezulu: I-Fasoracetam ingathola imikhiqizo ehlanzeka kakhulu ngezinqubo zokukhiqiza zokucwenga. Ukuhlanzeka okuphezulu kusho ukutholakala okungcono kwe-bioavailability kanye nokusabela okuncane okubi.
(2) Ukuphepha: Ucwaningo lubonise ukuthi i-fasoracetam ivame ukubekezelelwa kahle futhi ayibonisi imiphumela emibi ebalulekile uma isetshenziswa ngaphakathi kwemithamo enconyiwe.
(3) Ukuzinza: I-Fasoracetam inokuqina okuhle futhi ingagcina umsebenzi wayo kanye nomphumela ngaphansi kwezimo ezahlukene zokugcinwa.
Izicelo
I-Fasoracetam ivele njengenhlanganisela ethakazelisayo enamandla okuthuthukisa amakhono okuqonda, ikakhulukazi inkumbulo, ukunaka, nokufunda, futhi ingasetshenziswa njengesengezo sokudla. Lo mkhiqizo usebenza njengesithuthukisi senkumbulo ngokuvuselela ama-receptor e-glutamate e-metabolic. Emkhakheni wezinto eziphilayo, i-Fasoracetam isetshenziswa futhi njengesivimbeli esikhethiwe sokutadisha izinqubo zezinto eziphilayo ezifana nokusabalalisa amaseli kanye ne-apoptosis.












