I-Amino Tadalafil powder umkhiqizi we-CAS No.: 385769-84-6 98% ubumsulwa min. okwengeza izithako
Ividiyo Yomkhiqizo
Amapharamitha womkhiqizo
Igama lomkhiqizo | Amino Tadalafil |
Elinye igama | (6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A -Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR)-2-Amino-6-(benzo[d][1,3] ]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R ,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3 ,4-b]indole-1,4(6H,7H)-dione |
Inombolo ye-CAS. | 385769-84-6 |
Ifomula yamangqamuzana | I-C21H18N4O4 |
Isisindo samangqamuzana | 390.39 |
Ubumsulwa | 98.0% |
Ukubukeka | Impushana emhlophe ukuya kokumhlophe |
Isicelo | I-Dietary Supplement Raw Material |
Isingeniso somkhiqizo
I-Amino Tadalafil iyinhlanganisela entsha, ephuma ku-tadalafil, eya ngokuya idume emkhakheni we-erectile dysfunction (ED). Ihlanganisa i-amino acid ne-tadalafil, i-PDE5 inhibitor egunyazwe yi-FDA ngokuyinhloko esetshenziselwa ukwelapha i-ED. Isebenza ngokwandisa ukugeleza kwegazi epipini, okuvumela amadoda ukuthi afinyelele futhi agcine ukuqhanyelwa. Ngakolunye uhlangothi, ama-amino acid adlala indima ebalulekile emisebenzini ehlukahlukene yomzimba, okuhlanganisa ukukhiqizwa kwamaprotheni, okuyizici zokwakha izicubu nezitho. Inhlanganisela yalezi zithako ezimbili iklanyelwe ukuthuthukisa ukusebenza kahle kwe-Tadalafil ekwelapheni i-ED. Futhi i-amino Tadalafil inguqulo ethuthukisiwe enamandla angavamile, ethuthukisa ukusebenza nokuguquguquka kwalowo owandulelayo. Isakhiwo sayo samakhemikhali sihlala sifana neTadalafil, kodwa ngokusungulwa kwamaqembu e-amino, ithola izimfanelo eziyingqayizivele ezenza ivelele emhlabeni wemithi. Njenge-tadalafil, i-Amino Tadalafil isebenza ngokuvimbela i-phosphodiesterase 5 (PDE5), i-enzyme enesibopho sokudiliza i-cyclic guanosine monophosphate (cGMP) emzimbeni. I-cGMP iyinhlanganisela yemvelo ekhuthaza ukukhululeka kwemithambo yegazi, ngaleyo ndlela ikhulise ukugeleza kwegazi. Ngokuvimbela i-PDE5, i-amino Tadalafil iqinisekisa ukuqoqwa kwe-cGMP, ngaleyo ndlela ithuthukise i-vasodilation futhi ithuthukise ukujikeleza kwegazi. Ukwengeza, abacwaningi baye bahlola amandla ayo okusiza ukwelapha i-benign prostatic hyperplasia (BPH) ngokukhuthaza ukugeleza kwegazi ku-prostate.
Isici
(1) Ukuhlanzeka okuphezulu: I-Amino Tadalafil ingathola imikhiqizo ehlanzekile ngokusebenzisa izinqubo zokukhiqiza zokucwenga. Ukuhlanzeka okuphezulu kusho i-bioavailability engcono kanye nokusabela okungekuhle okumbalwa.
(2)Ukuphepha: Ukuphepha okuphezulu, ukusabela okungekuhle okumbalwa.
(3) Ukuzinza: I-Amino Tadalafil inokuzinza okuhle futhi ingagcina umsebenzi wayo kanye nomphumela ngaphansi kwezindawo ezahlukene nezimo zokugcina.
Izinhlelo zokusebenza
I-Amino Tadalafil iyi-PDE5 inhibitor enemiphumela efanayo yezemithi njenge-tadalafil. Ngokuhlanganisa ama-amino acid ne-tadalafil, i-amino Tadalafil kucatshangwa ukuthi iphumelela kakhulu ekwelapheni ukungasebenzi kahle kwe-erectile kune-tadalafil yodwa. Ama-amino acid angasiza ukuthuthukisa ukujikeleza kwegazi futhi asekele ukusebenza kahle okuphelele kwemithi. Ngaphezu kwalokho, ingathuthukisa izimpawu ze-erectile dysfunction (ED) ngokuvimbela umsebenzi we-PDE5 enzyme ukukhuthaza ukugeleza kwegazi ezithweni zesilisa zokuzala. Uma kuqhathaniswa ne-tadalafil, i-amino Tadalafil i-metabolized kancane kancane emzimbeni futhi ingase ikhiqize imiphumela ehlala isikhathi eside. Lokhu kunikeza i-amino Tadalafil amandla amakhulu ekwelapheni i-ED.