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umkhiqizo

I-Amino Tadalafil powder umkhiqizi we-CAS No.: 385769-84-6 98% ubumsulwa min.okwengeza izithako

Incazelo emfushane:

I-Amino Tadalafil iyinhlanganisela efana ne-Tadalafil, namanye amaqembu asebenzayo esakhiweni sayo athathelwa indawo ngamaqembu ama-amino.


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Amapharamitha womkhiqizo

Igama lomkhiqizo

Amino Tadalafil

Elinye igama

(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A -Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR)-2-Amino-6-(benzo[d][1,3] ]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R ,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3 ,4-b]indole-1,4(6H,7H)-dione

Inombolo ye-CAS.

385769-84-6

Ifomula yamangqamuzana

I-C21H18N4O4

Isisindo samangqamuzana

390.39

Ubumsulwa

98.0%

Ukubukeka

Impushana emhlophe ukuya kokumhlophe

Isicelo

I-Dietary Supplement Raw Material

Isingeniso somkhiqizo

I-Amino Tadalafil iyinhlanganisela efana ne-Tadalafil, namanye amaqembu asebenzayo esakhiweni sayo athathelwa indawo ngamaqembu ama-amino.I-PDE5 inhibitor futhi inemiphumela ye-pharmacological efana ne-Tadalafil.Isetshenziselwa ikakhulukazi ukwelashwa kwe-male erectile dysfunction (ED).Uma kuqhathaniswa ne-Tadalafil, i-Amino Tadalafil inezinga elincane le-metabolic emzimbeni, futhi ngaleyo ndlela ingaba nomphumela ohlala isikhathi eside.

Isici

(1) Ukukhetha okuphezulu: I-Amino Tadalafil inokukhetha okuphezulu kwe-PDE5, enobudlelwane obuphakeme kakhulu be-PDE5 kunamanye ama-subtypes e-PDE.Lokhu kusho ukuthi i-Amino Tadalafil ingavimbela ngokuphumelelayo umsebenzi we-enzyme ye-PDE5, ikhuthaze ukugeleza kwegazi ezingxenyeni zokuzala zesilisa futhi ithuthukise izimpawu ze-erectile dysfunction (ED).

(2) Umphumela ohlala isikhathi eside: I-Amino Tadalafil inezinga elincane le-metabolism emzimbeni, elivumela ukuthi likhiqize umphumela omude we-pharmacological, ohlala emahoreni angu-36.Lokhu kwenza i-Amino Tadalafil ibe yisidakamizwa sokwelapha se-ED eside, esingadingi ukuthathwa njalo.

(3) Imiphumela emibi embalwa: I-Amino Tadalafil inemiphumela emibi embalwa uma iqhathaniswa ne-Tadalafil, njengekhanda elibuhlungu, nokungahambi kahle kwamathumbu.Ngenxa yokukhethwa kwayo okuphezulu, i-Amino Tadalafil ingagwema ngokuphumelelayo ukusebenzisana namanye ama-subtypes e-PDE, ukunciphisa izehlakalo zemiphumela emibi.

(4) Amathemba ohlelo olubanzi: Ngaphezu kokwelapha i-ED, i-Amino Tadalafil ingase isetshenziselwe ukwelapha ezinye izifo ezifana ne-pulmonary arterial hypertension.Lokhu kwenza i-Amino Tadalafil ibe nethuba elibanzi lokufaka isicelo esikhathini esizayo.

Izinhlelo zokusebenza

I-Amino Tadalafil iyinhlanganisela eyakhiwe eminyakeni yamuva, enesakhiwo esifana ne-Tadalafil, kodwa amanye amaqembu esakhiweni sawo athathelwa indawo ngamaqembu ama-amino.Njengamanje, i-Amino Tadalafil ayizange ivunyelwe ukusetshenziswa kwezokwelapha, ngakho-ke ukusetshenziswa kwayo emkhakheni wezokwelapha kulinganiselwe.Kodwa-ke, ezinye izifundo zibonise ukuthi le nhlanganisela inamandla amakhulu okusetshenziswa.

I-Amino Tadalafil iyi-PDE5 inhibitor, enomphumela ofanayo we-pharmacological njenge-Tadalafil.Ingathuthukisa izimpawu ze-erectile dysfunction (ED) ngokukhuthaza ukugeleza kwegazi ezithweni zabesilisa zokuzala ngokuvimbela umsebenzi we-PDE5 enzyme.Uma kuqhathaniswa ne-Tadalafil, i-Amino Tadalafil inezinga elincane le-metabolism emzimbeni, elingase libe nomphumela ohlala njalo.Lokhu kwenza i-Amino Tadalafil ibe namandla amakhulu ekwelapheni i-ED.

Ngaphezu kwalokho, i-Amino Tadalafil ingasetshenziswa futhi ukwelapha ezinye izifo, njenge-pulmonary arterial hypertension.Olunye ucwaningo luye lwabonisa ukuthi i-PDE5 inhibitors inganweba imithambo yegazi yamaphaphu, ngaleyo ndlela ithuthukise izimpawu zeziguli ezine-pulmonary arterial hypertension.Ngenxa yokuthi i-Amino Tadalafil inomphumela ofanayo we-pharmacological njenge-Tadalafil, ingase isetshenziselwe ukwelapha i-pulmonary arterial hypertension.

Sekukonke, i-Amino Tadalafil inamandla amakhulu wokufaka isicelo, kodwa ukuhlolwa okwengeziwe kwemitholampilo kuyadingeka ukuze kunqunywe ukuphepha nokusebenza kwayo.Uma lezi zivivinyo ziveza imiphumela emihle, i-Amino Tadalafil ingase ibe umuthi omusha wokwelapha i-ED kanye ne-pulmonary arterial hypertension, ehlinzeka ngezinketho zokwelashwa ezengeziwe kodokotela basemtholampilo neziguli.


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