isibhengezo_sekhasi

umkhiqizo

Umkhiqizi wempuphu ye-Aniracetam Inombolo ye-CAS: 72432-10-1 Ubumsulwa obungu-99% bezithako ezengeziwe

Incazelo emfushane:

I-Aniracetam iyinhlanganisela yokwenziwa, enye yamakhemikhali e-hydroxyphenyl lacetamide heterocyclic, eyingxenye yezithuthukisi zomsebenzi wobuchopho kanye nama-neuroprotective agents. Isebenza ezingxenyeni zamaseli obuchopho (ama-neurons) abizwa ngokuthi ama-AMPA receptors.


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Ividiyo Yomkhiqizo

Amapharamitha Omkhiqizo

igama lomkhiqizo

1-(4-METHOXYBENZOYL)-2-PYRROLIDINONE; 1-(4-methoxybenzoyl)pyrrolidin-2-one;Aniracetam

Elinye igama

I-Aniracetam

Inombolo ye-CAS

72432-10-1

ifomula yama-molecule

C12H13NO3

isisindo sama-molecule

219.23

ubumsulwa

99%

Ukubukeka

Impuphu emhlophe

Ukupakisha

25kg/isigubhu

Isicelo

i-nootropic esezingeni eliphezulu

Isingeniso somkhiqizo

I-Aniracetam iyinhlanganisela yokwenziwa, enye yama-compound e-hydroxyphenylacetamide heterocyclic, okuyi-enhancer function function kanye ne-neuroprotective agent. Yaziwa ngekhono layo lokuthuthukisa inkumbulo, ukugxilisa ingqondo, kanye nomsebenzi wokuqonda jikelele. Yasungulwa ngawo-1970, i-Aniracetam yasheshe yathandwa ngenxa yezakhiwo zayo ezihlukile. Kukholakala ukuthi ithuthukisa ukuxhumana phakathi kwama-neurons ebuchosheni, ngaleyo ndlela ithuthukise izinqubo zokuqonda. Isebenza ikakhulukazi ezingxenyeni zamaseli obuchopho (ama-neurons) abizwa ngokuthi ama-AMPA receptors. Ama-AMPA receptors asiza izimpawu ukuthi zihambe ngokushesha phakathi kwama-neurons, okungathuthukisa inkumbulo, ukufunda, kanye nokukhathazeka. Indlela eqondile yokusebenza kwe-Aniracetam ukuthi isebenza kuma-receptor ahlukahlukene e-neurotransmitter ebuchosheni, njenge-acetylcholine kanye nama-dopamine receptors. Ngokuguqula la ma-receptor, kucatshangwa ukuthi i-Aniracetam yandisa ukukhululwa kanye nokutholakala kwama-neurotransmitter, ngaleyo ndlela ithuthukise ukusebenza kokuqonda.

Isici

(1) Ubumsulwa obuphezulu: I-Aniracetam ingaba umkhiqizo omsulwa kakhulu ngezinqubo zokukhiqiza ezicwengisisiwe. Ubumsulwa obuphezulu busho ukutholakala okungcono kwe-bioavailability kanye nokusabela okuncane okubi.

(2) Ukusabela okungekuhle okuphansi: ukuphepha okuphezulu, ukusabela okungekuhle okumbalwa, ukusabela okungekuhle okusobala ngisho noma kusetshenziswa isikhathi eside. Kodwa udinga ukunaka umthamo kanye nokungezwani komzimba.

(3) Ukuzinza: I-Aniracetam izinzile kahle futhi ingagcina umsebenzi wayo kanye nomphumela ngaphansi kwezimo ezahlukene zokugcinwa.

Izicelo

I-Aniracetam iyisithuthukisi somsebenzi wobuchopho esiphephile nesisebenzayo kanye nesivikela imizwa esinemiphumela ebalulekile ekuthuthukiseni inkumbulo, ikhono lokufunda kanye nezimpawu zokucindezeleka. Izifundo eziningi zikhombisile ukuthi i-Aniracetam ingathuthukisa ukwakheka kwenkumbulo yesikhathi esifushane neside, okuwusizo kubantu abafuna ukuthuthukisa amakhono abo okufunda. Esinye isici esithakazelisayo se-Aniracetam amandla ayo okuthuthukisa ubuhlakani. Abasebenzisi abaningi babika ukwanda kokucabanga okuhlukene, amakhono athuthukisiwe okuxazulula izinkinga, kanye nokugeleza kwemibono okushelelayo. Lokhu kungaba usizo kubantu abasemisebenzini yokudala noma kunoma ubani ofuna ukusebenzisa amandla akhe okudala.


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