Umkhiqizi wempuphu ye-Coluracetam Inombolo ye-CAS: 135463-81-9 99% ubumsulwa obuncane bezithako ezengeziwe
Ividiyo Yomkhiqizo
Amapharamitha Omkhiqizo
| Igama lomkhiqizo | I-Coluracetam |
| Elinye igama | I-MKC-231; 2-oxo-N-(5,6,7,8-tetrahydro-2,3-dimethyl-furo[2,3-b]quinolin-4-yl)-1-pyrrolidineacetamide |
| Inombolo ye-CAS | 135463-81-9 |
| Ifomula yama-molecule | C19H23N3O3 |
| Isisindo sama-molecule | 341.4 |
| Ubumsulwa | 99.0% |
| Ukubukeka | Impuphu emhlophe |
| Isicelo | Isengezo Sokudla Izinto Ezingavuthiwe |
Isingeniso somkhiqizo
I-Coluracetam, ilungu lomndeni we-racemate wama-nootropic compounds, aziwa nangokuthi i-MKC-231, iyinhlanganisela ye-nootropic enemiphumela yokuthuthukisa ingqondo kanye nokuvikela imizwa. I-Coluracetam isebenza ngokuguqula uhlelo lwe-cholinergic. Kucatshangwa ukuthi ikhulisa amazinga e-acetylcholine, i-neurotransmitter ebalulekile ebuchosheni ehlobene kakhulu nokufunda kanye nemisebenzi yememori. I-Coluracetam yenza lokhu ngokwandisa inani kanye nomsebenzi wabathuthi be-choline uptake, ngaleyo ndlela ithuthukise ukukhishwa kwe-acetylcholine futhi ithuthukise ukusayinwa phakathi kwama-neurons. Ezinye izifundo zokuhlola zakuqala kanye nezilwane ziphakamisa ukuthi i-Coluracetam inemiphumela engaba khona yokuvikela imizwa kanye nokuthuthukisa ingqondo. Ezinye izifundo zithole ukuthi i-Coluracetam inomphumela othile wokuthuthukisa ekulimaleni kwememori kumamodeli e-AD.
Isici
(1) Ukuhlanzeka okuphezulu: I-Coluracetam ilungiswa kusetshenziswa izinqubo zokukhipha nokukhiqiza ezithuthukisiwe ukuqinisekisa ukuhlanzeka okuphezulu. Lokhu kuhlanzeka okuphezulu kusiza ekuthuthukiseni ukutholakala kwezinto eziphilayo kanye nokunciphisa ukwenzeka kwemiphumela emibi.
(2) Ukuphepha: I-Coluracetam ibhekwa njengephephile kubantu. Ucwaningo oluningi luye lwafakazela ukuthi inobuthi obuphansi kanye nemiphumela emibi emincane ngaphakathi kobubanzi bomthamo obunconywayo.
(3) Ukuzinza: Amalungiselelo e-Coluracetam abonisa ukuzinza okuhle kakhulu futhi angagcina umsebenzi wawo kanye nokusebenza kahle ngaphansi kwezimo ezahlukene zokugcinwa. Lokhu kuzinza kuqinisekisa ukusebenza okuzinzile nokuthembekile isikhathi eside.
Izicelo
I-Coluracetam okwamanje isetshenziswa ezinhlotsheni ezahlukene zokusebenza futhi ikhombisa ithemba elikhulu lesikhathi esizayo. Isetshenziswa ngokuyinhloko njengesengezo sokudla esithuthukisa ingqondo futhi ifunwa ngabantu abafuna ukuthuthukisa inkumbulo, ukugxilisa ingqondo, kanye namakhono okufunda. Ikhono lale nhlanganisela lokuguqula uhlelo lwe-cholinergic kucatshangwa ukuthi lifaka isandla emiphumeleni yalo yokuthuthukisa ingqondo. Ngaphezu kwalokho, ucwaningo luphakamisa ukuthi i-Coluracetam ingaba nezakhiwo zokuvikela izinzwa ezingasiza ekuvimbeleni ukwehla kwengqondo okuhlobene nokuguga futhi isekele impilo yobuchopho iyonke.












