I-Compound 7P umkhiqizi we-powder CAS No.: 1890208-58-8 99% ubumsulwa min.okwengeza izithako
Amapharamitha womkhiqizo
Igama lomkhiqizo | Inhlanganisela 7P |
Elinye igama | I-Compound7P;2-[(2-methoxyphenyl)[(4-methylphenyl)sulfonyl]amino]-N-(4-methoxy-3-pyridinyl)acetamide; 2-(N-(2-methoxyphenyl)-4-methylphenylsulfonamido)-N-(4-methoxypyridin-3-yl)acetamide |
Inombolo ye-CAS. | 1890208-58-8 |
Ifomula yamangqamuzana | I-C22H23N3O5S |
Isisindo samangqamuzana | 441.51 |
Ubumsulwa | 99.0% |
Ukubukeka | Impushana emhlophe |
Isicelo | I-Nootropic |
Isingeniso somkhiqizo
I-Compound 7p yaboniswa ukuze ikhuthaze ukukhula kwama-axon e-GAP-43-positive kumodeli yezilwane yokulimala kwe-optic nerve, okuphakamisa ukuthi umsebenzi we-neurite outgrowth we-compound 7p in vitro uhumusha ekukhuthazeni ukuvuselelwa kwe-axon ku-vivo.I-Compound 7P powder iyimpushana emhlophe ukuya emhlophe ekhiqizwa njengenhlanganisela ye-tandem yokuhlonza i-thromboxane receptor antagonist inhibitors esebenza kabili.Ngempela, i-compound 7p ibonisa ukukhetha kwe-prostaglandin I2 synthase (PTGIS, CYP8A1) phezu kwe-thromboxane synthase (CYP5A1).I-nootropic yinoma iyiphi into esiza ukuthuthukisa ukusebenza kobuchopho, okuhlanganisa inkumbulo, ukugxilisa ingqondo, isimo sengqondo, ngisho nokuhlakanipha.Zingasukela emaqenjini athile okudla noma izinto kuye kwezinhlanganisela ezenziwe umuntu eziklanyelwe ukusiza ukusebenza kobuchopho nezinye izinzuzo.I-Nootropic compound 7P powder ikhuthaza ukuphuma kwe-Gap-43 ama-axon amahle, ngaleyo ndlela ikhuthaze ukuvuselelwa kwe-axonal ku-vivo.I-7p ehlanganisiwe yekhwalithi ephezulu iklanyelwe ukuthuthukisa ukusebenzisana, ukuthuthukisa isimo sengqondo nokusiza ukulwa nokukhathala.Iphinde ivimbele ukugcotshwa kobuchopho futhi isize ukulwa nokulimala kobuchopho okubangelwa ukuphuza utshwala.
Izinhlelo zokusebenza
Ama-Neurons ohlelweni lwezinzwa oluphakathi lwabantu abadala (CNS) ahluleka ukuvuselela ama-axon ngemva kokulimala, okuyingxenye echaza ukululama okungalungile kokusebenza ezigulini ezihlukumezekile kanye nezifo ze-neurodegenerative.I-Compound 7p, ethuthukisa ukuphuma kwe-neurite kuma-neuron athuthukisiwe atholakala ku-hippocampus, i-cerebral cortex, ne-retina, futhi ikhuthaza ukuvuselelwa kwenzwa ye-optic kumodeli yesilwane yokulimala kwenzwa ye-optic.Iphinde ikhulise ukusebenzisana, yelaphe ukulimala kobuchopho obuhlobene notshwala, futhi ivimbele i-oxidation ezungeze ubuchopho.Futhi kusiza ukuthuthukisa isimo somuntu nokulwa nokukhathala.Ukwengeza i-7P ehlanganisiwe ibonise umsebenzi ophezulu kakhulu ngokumelene nezimila zomlomo wesibeletho ngokwenza ngcono i-microstructure ngendlela encike kumthamo.Ukwenziwa ngcono okwengeziwe kwe-compound 7p kanye nokucaciswa kwendlela edala ngayo ukuvuselelwa kwe-axon ku-vivo kuzohlinzeka ngesizathu semizamo yesikhathi esizayo yokuqinisa amasu okwelapha.