I-5a-Hydroxy Laxogenin powder umkhiqizi we-CAS No.: 56786-63-1 98% ubumsulwa min.okwengeza izithako
Amapharamitha womkhiqizo
Igama lomkhiqizo | 5a-Hydroxy lxogenin |
Elinye igama | 5A-hydroxy lacosgenin |
Inombolo ye-CAS. | 56786-63-1 |
Ifomula yamangqamuzana | I-C27H42O5 |
Isisindo samangqamuzana | 446.62 |
Ubumsulwa | 98.0% |
Ukubukeka | Impushana emhlophe |
Ukupakisha | 1 kg/isikhwama 25kg/isigubhu |
Isicelo | Pharmaceutical Intermediate |
Isingeniso somkhiqizo
I-Laxogenin, eyaziwa nangokuthi i-5 α Hydroxy Laxogenin noma i-5a hydroxy Laxogenin ibizwa ngokuthi i-plant steroid ngoba isuka ku-Smilax Sieboldii, equkethe i-brassinosteroids.Isiqu esingaphansi komhlaba sesitshalo sase-Asia i-Smilax sieboldii siqukethe cishe u-0.06% we-laxogenin, okuwumthombo wayo wemvelo oyinhloko.I-Laxogenin iphinde itholakale kuma-bulb ka-anyanisi waseShayina (i-Allium genus) futhi iyinhlanganisela yezitshalo, ilungu elidume kakhulu leqembu lezinhlanganisela ezaziwa ngokuthi ama-brassinosteroids, afana ne-cholesterol etholakala kumahomoni ocansi omuntu.I-Rapeseed steroids ibonise imiphumela ye-anabolic, engathuthukisa ukusebenza komzimba womuntu ngezindlela ezihlukahlukene.Kodwa-ke, njengesitshalo esiyingqayizivele esivela kwamakhemikhali, i-laxogenin ingathinta izindlela ezahlukene emzimbeni.Ngaphezu kwalokho, okuphuma ku-laxogenin yemvelo kuvimbela i-enzyme (phosphodiesterase) ephula i-cAMP.Lokhu kuzonyusa amazinga e-cAMP, kuthuthukise ukuwohloka kwamafutha, futhi kuqalise ukulwa noma ukuphunyuka (okunozwelo).
Isici
(1) Sheshisa ukukhula kwezicubu ezithambile.
(2) Khulisa ukwakheka kwamaprotheni, okwenza kusebenze izinhlobo ezithile zamaprotheni emzimbeni futhi aqinisekise ukuthi umzimba wakho awephuli amaprotheni emisipha.Ngamaprotheni amaningi emisipha, umzimba wakho uzokwazi ukuthuthukisa ngokuphawulekayo ukusebenza kwawo.Uzolulama ngokushesha futhi ikhwalithi izoshesha.
(3) Ukubola ama-adipocyte.
Izinhlelo zokusebenza
I-5a-hydroxylaxogenin iyinhlanganisela ye-homologous ye-laxogenin futhi iyi-steroid yemvelo etholakala ezitshalweni eziningi eziluhlaza.Inomsebenzi we-anabolic/androgenic, ofana kakhulu ne-anavar yokwenziwa ye-metabolite ephumelelayo kakhulu.Kuyinhlanganisela ye-anabolic kakhulu engakhuthaza ukukhula kwezicubu ezithambile emzimbeni.Kuyinhlanganisela ethengiswa ngezindlela ezahlukahlukene njengesengezo sokumisa imisipha.Ingokwesigaba samahomoni ezitshalo abizwa nge-brassinosteroids, futhi ukwakheka kwawo kufana namahomoni e-steroid ezilwane.