isibhengezo_sekhasi

umkhiqizo

Umkhiqizi wempuphu yePramiracetam Inombolo ye-CAS: 68497-62-1 Ubumsulwa obungu-98% bezithako ezengeziwe

Incazelo emfushane:

I-Pramiracetam iyisidakamizwa sokuthuthukisa ukusebenza kahle kobuchopho se-pyrrolidone, okuwumuthi oyinhloko wezinzwa ongathuthukisa inkumbulo kanye nokulwa nokukhohlwa.


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Ividiyo Yomkhiqizo

Amapharamitha Omkhiqizo

Igama lomkhiqizo

I-Pramiracetam

Elinye igama

I-Amacetam;

I-N-[2-(Diisopropylamino)ethyl]-2-oxo-1-pyrrolidineacetamide;N-(2-(Bis(1-methylethyl)amino)ethyl)-2-oxo-1-pyrrolidineacetamide;

I-NeupraMir;

I-PraMistar;

ReMen;

I-Vinpotropil

Inombolo ye-CAS

68497-62-1

Ifomula yama-molecule

C14H27N3O2

Isisindo sama-molecule

269.38

Ubumsulwa

99.0%

Ukubukeka

Impuphu emhlophe ekristalu

Ukupakisha

25 kg/umgqomo

Isicelo

I-Nootropic

Isingeniso somkhiqizo

I-Pramiracetam iyingxenye yomndeni wemithi ye-nootropic eyaziwa ngezakhiwo zayo zokuthuthukisa ingqondo. iyinhlanganisela ye-nootropic ethathwe ku-Racetam, isithuthukisi sokuqonda esidumile. I-Pramiracetam ifana ngamakhemikhali ne-piracetam, i-piracetam yokuqala eyatholakala, kodwa kukholakala ukuthi inamandla kakhulu. Ukuze siqonde imiphumela ye-pramiracetam ekusebenzeni kwengqondo, kumele singene ngokujulile endleleni esebenza ngayo. I-Pramiracetam isebenza ngokushintsha i-acetylcholine ye-neurotransmitter ebuchosheni, okuholela ekwandeni komsebenzi we-cholinergic. Lo mthetho ungaholela ekukhulisweni kwenkumbulo, ukunakwa okwandisiwe, ukufunda okuthuthukisiwe, kanye namakhono okuqonda athuthukisiwe jikelele. Iphinde ivuselele ukukhishwa kwe-dopamine, i-neurotransmitter ephethe imizwa ejabulisayo, ngaleyo ndlela isize ekwandiseni isisusa nokugxila. I-Pramiracetam ixhunywe ekuthuthukisweni kokugxilisa ingqondo kanye nesikhathi sokunaka. Ngokwandisa ukugeleza kwegazi ebuchosheni kanye nokuvuselela ama-receptor e-cholinergic, ingasiza abantu ukuthi bagxile kunoma yimuphi umsebenzi isikhathi eside.

Isici

(1) Ukuhlanzeka okuphezulu: I-Pramiracetam ingathola imikhiqizo ehlanzeka kakhulu ngezinqubo zokukhiqiza zokucwenga. Ukuhlanzeka okuphezulu kusho ukutholakala okungcono kwe-bioavailability kanye nokusabela okuncane okubi.

(2) Ukuphepha: I-Praracetam ifakazelwe ukuthi iphephile emzimbeni womuntu.

(3) Ukuzinza: I-Pramiracetam izinzile kahle futhi ingagcina umsebenzi wayo kanye nomphumela ngaphansi kwezimo ezahlukene zokugcinwa.

Izicelo

I-Pramiracetam iyisengezo sokudla esinamandla se-nootropic esiyilungu lomndeni wezidakamizwa ze-racemate. I-Pramiracetam ithuthukisa ukuntuleka kwengqondo okuhambisana nokulimala kobuchopho okubuhlungu. Ngaphezu kwalokho, i-pramiracetam iyisithibi esithile se-prolyl endopeptidase. I-Pramiracetam idlala indima ebalulekile ekufundeni kwendawo kanye nenkumbulo futhi ibhekwa njengesithuthukisi senkumbulo, esinamandla kakhulu kune-piracetam. I-Pramiracetam ithuthukisa ukusebenza kwengqondo ebuchosheni ngokwandisa ukukhishwa kwe-neurotransmitter acetylcholine. Iphinde ikhulise inani kanye nokuxhumana kwama-neurons, ikhuthaze ukukhula nokulungiswa kwe-neuronal. I-Pramiracetam ingakhulisa futhi izinga lokuguqulwa kobuchopho futhi ikhulise ukugeleza kwegazi kobuchopho, ngaleyo ndlela ithuthukise ukunikezwa komoya-mpilo nezakhamzimba ebuchosheni.


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